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Publications récentes


-Tether influence on the binding properties of tRNALys3 ligands designed by a fragment based approach.

R. Moumné, V. Larue, B. Seijo, T. Lecourt, L. Micouin and C. Tisné,

Org. Biomol. Chem. 2010, 8, 1154-1159

-Copper-Catalyzed Ring-Opening of Polycyclic Hydrazines With Trialkylaluminium Reagents and SimplePhos Ligands.

L. Palais, C. Bournaud, L. Micouin, A. Alexakis,

Chem. Eur. J. 2010, 16, 2567-2573.

-Direct Synthesis of 1,4-Disubstituted-5-alumino-1,2,3-triazoles By a Copper-Catalyzed Cycloaddition of Organic Azides and Mixed-Aluminum acetylides.

Y. Zhou, T. Lecourt, L. Micouin,

Angew. Chem. Int. Ed. 2010, 49, 2607-2610.

-Fluorinated Diaminocyclopentanes as Chiral Sensitive NMR Probes of RNA Structure.

R. Moumné, M. Pasco, E. Prost, T. Lecourt, L. Micouin, C. Tisné,

J. Am. Chem. Soc. 2010, 132, 13111-13113.

-Rh(II) carbene-promoted activation of the anomeric C-H bond of carbohydrates : a stereospecific entry towards α- and β-ketopyranosides.

M. Boultadakis-Arapinis, P. Lemoine, S. Turcaud, L. Micouin, T. Lecourt,

J. Am. Chem. Soc. 2010, 132, 15477-15479.

-Rhodium(II) carbene-mediated modification of 2-deoxystreptamine surrogates.

A. Blond, R. Moumné, G. Bégis, M. Pasco, T. Lecourt, L. Micouin

Tetrahedron Lett. 2011, 52, 3201-3203.

-Stereoselective synthesis of fluorinated 1,3-cis-diaminocyclopentanes.

M. Pasco, R. Moumné, T. Lecourt, L. Micouin

J. Org. Chem. 2011, 76, 5237-5142.

-Chemodivergent synthesis of 7-Aryl/alkyl-6-hydroxy-1,4-oxazepan-5-ones and 2-[Aryl/alkyl(hydroxy)methyl]morpholin-3-ones from a common epoxyamide precursor.

D. M. Apraicio, J. L. Teran, L. F. Roa, D. Gnesso, J. R. Juarez, M. L. Orea, A. Mendoza, M. Flores-Alamo, L. Micouin

Synthesis, 2011, 2310-2320.

-Rh(II) Carbene-Mediated Synthesis of Methyl α- and β-Ketopyranosides : Preparation of Carbene Precursors, Quaternarization of the Anomeric Position, and Ring Opening of γ-Lactone.

M. Boultadakis-Arapinis, C. Lescot, L. Micouin, T. Lecourt

Journal of Carbohydrate Chemistry, 2011, 30:7-9, 587-604.

-Direct Synthesis of Polysubstituted Aluminoisoxazoles and Pyrazoles by a Metalative Cyclization.

O. Jackowski, T. Lecourt, L. Micouin

Org. Lett., 2011, 13, 5664-5667

-Fragment-based design of small RNA binders : promising developments and contribution of NMR.

R. Moumné, M. Catala, V. Larue, L. Micouin, C. Tisné

Biochimie 2012, 94, 1607-1619

-Investigation of RNA-ligand interaction by 19F NMR spectroscopy using fluorinated probes.

T. Lombès, R. Moumné, V. Larue, E. Prost, M. Catala, T. Lecourt, F. Dardel, L. Micouin, C. Tisné,

Angew. Chem. Int. Ed. 2012, 51, 9530-9534

-Gram-Scale Quaternarization of the Anomeric Position of Carbohydrates : Dramatic Effects of Molecular Sieves on Rh(II)-Mediated Decomposition of Diazo sugars.

M. Boultadakis Arapinis, C. Lescot, L. Micouin, T. Lecourt,

Synthesis 2012, 44, 3731-3734

-Recent developments in the synthesis 1,4,5-trisubstituted triazoles

Mignani, S. ; Zhou, Y. ; Lecourt, T. ; Micouin,

L. Topics in Heterocyclic Chemistry, 2012, Vol. 28, 185-232.

-2,3-Diazabicyclo[2.2.1]hept-5-ene-2,3-dicarboxylic Acid, 2,3-Diethyl Ester,

B. A. Bhanu Prasad, S. R. Gilbertson, T. Lombès , L. Micouin

in eEROS, John Wiley & Sons, UK, 2012, DOI : 10.1002/047084289X.rn01437

-Carbene-Mediated Functionalization of the Anomeric C-H Bond of Carbohydrates : Scope and Limitations

M. Boultadakis Arapinis, E. Prost, V. Gandon, P. Lemoine, S. Turcaud, L. Micouin, T. Lecourt,

Chem. Eur. J. 2013, 19, 6052-6066

-Functionalization of the anomeric C-H bond of carbohydrates : old strategies and new opportunities

M. Boultadakis Arapinis, C. Lescot, S. Turcaud, L. Micouin, T. Lecourt,

Synlett 2013, 2477-2491

-Modular access to N-substituted cis-3,5-diaminopiperidines

A. Blond, P. Dockerty, R. Álvarez, S. Turcaud, T. Lecourt, L. Micouin,

J. Org. Chem. 2013, 78, 12226-12242

-Electronic effects in Carbene-Mediated C-H Bond functionalization : An Experimental and Theoretical Study

M. Boultadakis-Arapinis, V. Gandon, E. Prost, L. Micouin, T. Lecourt,

Adv. Synth. Catal. 2014, 356, 2493-2505

-The design of RNA binders : targeting the HIV replication cycle as a case study

A. Blond, E. Ennifar, C. Tisné, L. Micouin,

ChemMedChem 2014, 9, 1982-1996

-The reaction of dimethylalkynylaluminum reagents with trimethylsilyldiazomethane : original reactivity leading to new silylated alkynylhydrazones

R. Kumar, S. Turcaud, L. Micouin,

Org.Lett. 2014, 16, 6192-6195



Publications récentes
-Stereoselective Transformations of meso-Bicyclic Hydrazines : a Versatile Access to Functionalized Amino-Cyclopentanes. C. Bournaud, F. Chung, A. Perez Luna, M. Pasco, G. Errasti, T. Lecourt, L. Micouin,
Synthesis 2009, 869-887.
-  Desymmetrization of hydrazinocyclohexadienes : a new approach for the synthesis of polyhydroxylated aminocyclohexanes.
G. Errasti, C. Koundé, T. Lecourt, O. Mirguet, L. Micouin,
Org. Lett. 2009, 11, 912-915.
-  NMR-guided fragments (...)




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